Achievements

Name: Masayuki Inoue

Original papers

  • "Installation of O-Heterocycles to N-Heteroarenes via an Et3B/O2-mediated Radical Reaction of a-Alkoxy and a-Alkoxyacyl Tellurides"
    Kuwana, D.; Ovadia, B.; Kamimura, D.; Nagatomo, M.; *Inoue M.
    Asian J. Org. Chem.,2019, 8, XX-XX
  • "Construction of a 6/5/9-membered Tricyclic Structure of Cladiellins via Radical-polar Crossover Reaction"
    Nagatomo, M.; Fujimoto, Y.; Masuda, K.; *Inoue M.
    J. Antibiot.,2019
  • "Convergent Synthesis of Taxol Skeleton via Decarbonylative Radical Coupling Reaction"
    Matoba, H.; Watanabe, T.; Nagatomo, M.; *Inoue M.
    Org. Lett.,2018, 20, 7554-7557
  • "Convergent Total Synthesis of Asimicin via Decarbonylative Radical Dimerization"
    Kawamata, T.; Yamaguchi, A.; Nagatomo, M.; *Inoue M.
    Chem. Eur. J.,2018, 24, 18907 -18912
  • "Total Synthesis and Biological Evaluation of 19-Hydroxysarmentogenin-3-O-a-L-rhamnoside, Trewianin, and Their Aglycons"
    Urabe, D.; Nakagawa, Y.; Mukai, K.; Fukushima, K.; Aoki, N.; Itoh, H.; Nagatomo, M.; *Inoue, M.
    J. Org. Chem.,2018, 83, 13888-13910
  • "Target Identification of Yaku’amide B and Its Two Distinct Activities against Mitochondrial FoF1-ATP Synthase"
    Kitamura, K.; Itoh, H.; Sakurai, K.; Dan, S.; *Inoue M.
    J. Am. Chem. Soc.,2018, 140, 12189-12199
  • "Construction of a Pentacyclic Ring System of Isoryanodane Diterpenoids by SmI2-mediated Transannular Cyclization"
    Koshimizu, M.; Nagatomo, M.; *Inoue, M.
    Tetrahedron,2018, 74, 3384-3390
  • "A Three-Component Coupling Approach to the ACE-Ring Substructure of C19-Diterpene Alkaloids"
    Minagawa, K.; Urabe, D.; *Inoue, M.
    J. Antibiot.,2018, 71, 326-332
  • "Synthesis of the Tetracyclic Structure of Batrachotoxin Enabled by Bridgehead Radical Coupling and Pd/Ni-Promoted Ullmann Reaction"
    Sakata, K.; Wang, Y.; Urabe, D.; *Inoue, M.
    Org. Lett.,2018, 20, 130-133
  • "Total Synthesis of Resiniferatoxin Enabled by Radical-Mediated Three-Component Coupling and 7-endo Cyclization"
    Hashimoto, S.; Katoh, S.; Kato, T.; Urabe, D.; *Inoue, M.
    J. Am. Chem. Soc.,2017, 139, 16420-16429
  • "Unified Total Synthesis of Polyoxin J, L, and Fluorinated Analogues on the Basis of Decarbonylative Radical Coupling Reactions"
    Fujino, H.; Nagatomo, M.; Paudel, A.; Panthee, S.; Hamamoto, H.; Sekimizu, K.; *Inoue, M.
    Angew. Chem., Int. Ed.,2017, 56, 11865-11869

Review

  • 「Comprehensive Structure-Activity Relationship Studies of Macrocyclic Natural Products Enabled by Their Total Syntheses」 Itoh, H.; *Inoue M., Chem. Rev., 119, XX-XX,2019

Conference

  • Pharmaron Lecture, Peking University Shenzhen Graduate School
    "Total Synthesis and Biological Evaluation of Complex Natural Products", 招待講演
    Inoue, M.
    4/19/2019, Shenzhen, China
  • Southern University of Science and Technology
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    4/18/2019, Shenzhen, China
  • 6th UK-Japan Conference on Asymmetric Catalysis
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    11/6/2018, Fukuoka, Japan
  • International Symposium on Frontiers of Natural and Biomimetic Drugs on “Natural Product Synthesis”
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    10/18/2018, Beijing, China
  • 22nd International Conference on Organic Synthesis (22-ICOS)
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    9/20/2018, Florence, Italy
  • 24th Conference on Isoprenoids
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    9/11/2018, Białystok, Poland
  • 256th ACS National Meeting (JOC Lectureship)
    "Total Synthesis and Biological Evaluation of Peptide Natural Products", 招待講演
    Inoue, M.
    8/19/2018, Boston, USA
  • Novartis Lectureship
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    6/21/2018, Toronto, Canada
  • Swiss Chemical Society Lectureship
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    5/7/2018-5/15/2018, Zurich, Bern, Fribourg, Genève, Lausanne, Basel, Switzerland
  • ACP Lectureship, Department of Chemistry, National Tsing Hua University
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    1/24/2018, Hsinchu, Taiwan
  • ACP Lectureship, Institute of Biotechnology and Pharmaceutical Research
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    1/23/2018, Taipei, Taiwan
  • ACP Lectureship, Institute of Chemistry, Academia Sinica
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    1/22/2018, Taipei, Taiwan

Award

  • 「The Journal of Organic Chemistry Outstanding Publication of the Year Award Lectureship」
    受賞者:Inoue, M.
    贈呈元:
    受賞日:
  • 「Swiss Chemical Society Lectureship Award 2017/2018」
    受賞者:Inoue, M
    贈呈元:
    受賞日:

Conference Management

  • 国際会議, Local Host, ACS on Campus, Tokyo, Japan, 6/15/2018