Achievements

Name: Masayuki Inoue

Original papers

  • "Total Synthesis of 1-Hydroxytaxinine"
    Imamura, Y.; Yoshioka, S.; Nagatomo, M.; *Inoue, M.
    Angew. Chem., Int. Ed., 2019, 58, 12159-12163
  • "Total Synthesis of 5-epi-Eudesm-4(15)-ene-1β,6β-diol via Decarbonylative Radical Coupling Reaction"
    Kuwana, D.; Nagatomo, M.; *Inoue, M.
    Org. Lett., 2019, 21, 7619-7623
  • "Biological Effects of a Simplified Synthetic Analogue of Ion-Channel-Forming Polytheonamide B on Plasma Membrane and Lysosomes"
    Xue, Y.-W.; Hayata, A.; Itoh, H.; *Inoue, M.
    Chem. Eur. J., 2019, 25, 15198-15204
  • "Total Synthesis of Talatisamine"
    Kamakura, D.; Todoroki, H.; Urabe, D.; Hagiwara, K.; *Inoue, M.
    Angew. Chem., Int. Ed., 2020, 59, 479-486
  • "Solid-Phase Total Synthesis of Yaku'amide B Enabled by Traceless Staudinger Ligation"
    toh, H.; Miura, K.; Kamiya, K.; Yamashita, T.; *Inoue, M.
    Angew. Chem., Int. Ed. , 2020, 59, 4564-4571
  • "Installation of O-Heterocycles to N-Heteroarenes via an Et3B/O2-mediated Radical Reaction of a-Alkoxy and a-Alkoxyacyl Tellurides"
    Kuwana, D.; Ovadia, B.; Kamimura, D.; Nagatomo, M.; *Inoue M.
    Asian J. Org. Chem., 2019, 8, 1088-1091
  • "Construction of a 6/5/9-membered Tricyclic Structure of Cladiellins via Radical-polar Crossover Reaction"
    Nagatomo, M.; Fujimoto, Y.; Masuda, K.; *Inoue M.
    J. Antibiot.,2019
  • "Convergent Synthesis of Taxol Skeleton via Decarbonylative Radical Coupling Reaction"
    Matoba, H.; Watanabe, T.; Nagatomo, M.; *Inoue M.
    Org. Lett.,2018, 20, 7554-7557
  • "Convergent Total Synthesis of Asimicin via Decarbonylative Radical Dimerization"
    Kawamata, T.; Yamaguchi, A.; Nagatomo, M.; *Inoue M.
    Chem. Eur. J.,2018, 24, 18907 -18912
  • "Total Synthesis and Biological Evaluation of 19-Hydroxysarmentogenin-3-O-a-L-rhamnoside, Trewianin, and Their Aglycons"
    Urabe, D.; Nakagawa, Y.; Mukai, K.; Fukushima, K.; Aoki, N.; Itoh, H.; Nagatomo, M.; *Inoue, M.
    J. Org. Chem.,2018, 83, 13888-13910
  • "Target Identification of Yaku’amide B and Its Two Distinct Activities against Mitochondrial FoF1-ATP Synthase"
    Kitamura, K.; Itoh, H.; Sakurai, K.; Dan, S.; *Inoue M.
    J. Am. Chem. Soc.,2018, 140, 12189-12199
  • "Construction of a Pentacyclic Ring System of Isoryanodane Diterpenoids by SmI2-mediated Transannular Cyclization"
    Koshimizu, M.; Nagatomo, M.; *Inoue, M.
    Tetrahedron,2018, 74, 3384-3390
  • "A Three-Component Coupling Approach to the ACE-Ring Substructure of C19-Diterpene Alkaloids"
    Minagawa, K.; Urabe, D.; *Inoue, M.
    J. Antibiot.,2018, 71, 326-332
  • "Synthesis of the Tetracyclic Structure of Batrachotoxin Enabled by Bridgehead Radical Coupling and Pd/Ni-Promoted Ullmann Reaction"
    Sakata, K.; Wang, Y.; Urabe, D.; *Inoue, M.
    Org. Lett.,2018, 20, 130-133
  • "Total Synthesis of Resiniferatoxin Enabled by Radical-Mediated Three-Component Coupling and 7-endo Cyclization"
    Hashimoto, S.; Katoh, S.; Kato, T.; Urabe, D.; *Inoue, M.
    J. Am. Chem. Soc.,2017, 139, 16420-16429
  • "Unified Total Synthesis of Polyoxin J, L, and Fluorinated Analogues on the Basis of Decarbonylative Radical Coupling Reactions"
    Fujino, H.; Nagatomo, M.; Paudel, A.; Panthee, S.; Hamamoto, H.; Sekimizu, K.; *Inoue, M.
    Angew. Chem., Int. Ed.,2017, 56, 11865-11869

Review

  • 「生物活性カルデノリド類の収束的全合成」 占部大介, *井上将行, 有機合成化学協会誌, 2019, 77, 452-462
  • 「Full Solid-Phase Total Synthesis of Macrocyclic Natural Peptides Using Four-Dimensionally Orthogonal Protective Groups」 Itoh, H.; *Inoue, M., Org. Biomol. Chem., 2019, 17, 6519-6527
  • 「Comprehensive Structure-Activity Relationship Studies of Macrocyclic Natural Products Enabled by Their Total Syntheses」 Itoh, H.; *Inoue M., Chem. Rev., 2019, 119, 10002-10031

Conference

  • Department of Chemistry, University of South Florida
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    11/25/2019, Tampa, FL, USA
  • (Tarrant Distinguished Visiting Professorship), Department of Chemistry, University of Florida
    "Radical-Based Approach for Synthesis of Complex Natural Products (2)", 招待講演
    Inoue, M.
    11/19/2019, Gainesville, FL, USA
  • (Tarrant Distinguished Visiting Professorship), Department of Chemistry, University of Florida
    "Total Synthesis and Biological Evaluation of Peptide Natural Products", 招待講演
    Inoue, M.
    11/19/2019, Gainesville, FL, USA
  • (Tarrant Distinguished Visiting Professorship), Department of Chemistry, University of Florida
    "Radical-Based Approach for Synthesis of Complex Natural Products (1)", 招待講演
    Inoue, M.
    11/18/2019, Gainesville, FL, USA
  • Multidisciplinary Lecture Series in Life Sciences & Technology, The University of Tokyo
    "Total Synthesis and Biological Evaluation of Structurally Complex Natural Products", 招待講演
    Inoue, M.
    7/18/2019, Tokyo, Japan
  • Summer Program, Nanoscience Part I: Biotechnology, The University of Tokyo
    "Total Synthesis and Biological Evaluation of Structurally Complex Natural Products", 招待講演
    Inoue, M.
    7/17/2019, Tokyo, Japan
  • 47th Naito Conference, C-H Bond Activation and Transformation
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    7/3/2019, Sapporo, Japan
  • The 1st International Symposium on Hybrid Catalysis for Enabling Molecular Synthesis on Demand
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    5/31/2019, Tokyo, Japan
  • Pharmaron Lecture, Peking University Shenzhen Graduate School
    "Total Synthesis and Biological Evaluation of Complex Natural Products", 招待講演
    Inoue, M.
    4/19/2019, Shenzhen, China
  • Southern University of Science and Technology
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    4/18/2019, Shenzhen, China
  • 6th UK-Japan Conference on Asymmetric Catalysis
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    11/6/2018, Fukuoka, Japan
  • International Symposium on Frontiers of Natural and Biomimetic Drugs on “Natural Product Synthesis”
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    10/18/2018, Beijing, China
  • 22nd International Conference on Organic Synthesis (22-ICOS)
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    9/20/2018, Florence, Italy
  • 24th Conference on Isoprenoids
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    9/11/2018, Białystok, Poland
  • 256th ACS National Meeting (JOC Lectureship)
    "Total Synthesis and Biological Evaluation of Peptide Natural Products", 招待講演
    Inoue, M.
    8/19/2018, Boston, USA
  • Novartis Lectureship
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    6/21/2018, Toronto, Canada
  • Swiss Chemical Society Lectureship
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    5/7/2018-5/15/2018, Zurich, Bern, Fribourg, Genève, Lausanne, Basel, Switzerland
  • ACP Lectureship, Department of Chemistry, National Tsing Hua University
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    1/24/2018, Hsinchu, Taiwan
  • ACP Lectureship, Institute of Biotechnology and Pharmaceutical Research
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    1/23/2018, Taipei, Taiwan
  • ACP Lectureship, Institute of Chemistry, Academia Sinica
    "Radical-Based Approach for Synthesis of Complex Natural Products", 招待講演
    Inoue, M.
    1/22/2018, Taipei, Taiwan

Award

  • 「Tarrant Distinguished Visiting Professorship」
    受賞者:Inoue, M.
    贈呈元:University of Florida
    受賞日:
  • 「Oral Presentation Award」
    受賞者:Shimakawa, T.
    贈呈元:The 9th Junior International Conference on Cutting-Edge Organic Chemistry in Asia
    受賞日:9/25/2019
  • 「Poster Presentation Award」
    受賞者:Kuwana, D.
    贈呈元:27th International Society of Heterocyclic Chemistry Congress
    受賞日:9/6/2019
  • 「The Journal of Organic Chemistry Outstanding Publication of the Year Award Lectureship」
    受賞者:Inoue, M.
    贈呈元:
    受賞日:
  • 「Swiss Chemical Society Lectureship Award 2017/2018」
    受賞者:Inoue, M
    贈呈元:
    受賞日:

Collaborative Research

Conference Management

  • 国際会議, Local Host, ACS on Campus, Tokyo, Japan, 6/15/2018